Human SET domain containing (lysine methyltransferase) 7 in complex with inhibitor (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide

Target ID: 
SETD7
Deposition Date: 
Monday 12th March 2012
Families: 
Transferases
Related Diseases: 
MetabolismChromatin and epigenetics
Structure type: 
protein-ligand

Download Coordinates:

4E47
Authors: 
Walker JR, Ouyang H, Dong A, Fish P, Cook A, Barsyte D, Vedadi M, Tatlock J, Owen D, Bunnage M, Bountra C, Edwards AM, Arrowsmith CH, Brown PJ
Site: 
Toronto
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