Human euchromatic histone lysine methyltransferase 1, catalytic domain, in complex with inhibitor MS012

Target ID: 
EHMT1
Aliases: 
bA188C12.1DKFZp667M072Eu-HMTase1EUHMTASE1FLJ12879FP13812GLPKIAA1876KMT1DRP11-188C12.1
Deposition Date: 
Thursday 3rd November 2016
Families: 
Methyltransferases
Related Diseases: 
CancerChromatin and epigenetics
Structure type: 
protein-ligand

Download Coordinates:

5TTG
Authors: 
Dong A, Zeng H, Liu J, Xiong Y, Babault N, Jin J, Tempel W, Bountra C, Arrowsmith CH, Edwards AM, Wu H, Brown PJ
Site: 
Toronto
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