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Human histone-lysine N-methyltransferase SETDB1, triple Tudor domain, in complex with aryl triazole fragment
Target ID:
SETDB1Deposition Date:
Thursday 28th September 2017Families:
Methyl-lysine readersRelated Diseases:
Cancer and epigeneticsStructure type:
protein-ligandDownload Coordinates:
6AU2Authors:
Mader P, Mendoza-Sanchez R, Iqbal A, Dong A, Dobrovetsky E, Corless VB, Liew SK, Tempel W, Smil D, Dela Sena CC, Kennedy S, Diaz D, Holownia A, Vedadi M, Brown PJ, Santhakumar V, Bountra C, Edwards AM, Yudin AK, Arrowsmith CH